Abstract:
:The cyclization of N-Boc-α-alkylserines to corresponding β-lactones under Mitsunobu reaction conditions and the ring opening with heterocyclic amines (pyrrolidine, piperidine, morpholine and thiomorpholine) produced N-Boc-α-alkyl-β-(sec-amino)alanines. The removal of the Boc group gives di-hydrochlorides of non-protein amino acids.
journal_name
Amino Acidsjournal_title
Amino acidsauthors
Olma A,Lasota A,Kudaj Adoi
10.1007/s00726-011-1055-3subject
Has Abstractpub_date
2012-06-01 00:00:00pages
2525-8issue
6eissn
0939-4451issn
1438-2199journal_volume
42pub_type
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