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Synthesis of diacylamines and the preparation of alpha-amino-acylureas, a new type of alpha-amino acid derivatives.

Abstract：

:Sixteen new and one known unsymmetrical open-chain diacylamines were synthesized by sodium methoxide catalyzed acylation of amides with carboxylic esters and acylamino-carboxylic esters, or acylureas with acylamino-carboxylic esters and alpha-amino acid esters.

journal_name

Bioorg Med Chem Lett

journal_title

Bioorganic & medicinal chemistry letters

authors

Weisz I,Roboz J,Wolf I,Szabo J,Bekesi JG

doi

10.1016/s0960-894x(98)00593-9

subject

Has Abstract

pub_date

1998-11-17 00:00:00

pages

3241-4

issue

22

eissn

0960-894X

issn

1464-3405

pii

S0960894X98005939

journal_volume

8

pub_type

杂志文章

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