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5-Carboxamido-1,3,2-dioxaphosphorinanes, potent inhibitors of MTP.

Abstract：

:5-Carboxamido-1,3,2-dioxaphosphorinanes have been identified as potent inhibitors of microsomal triglyceride-transfer protein. The 1,3,2-dioxaphosphorine functionality acted as a neutral and stable replacement for piperidine and piperidine N-oxide.

journal_name

Bioorg Med Chem Lett

journal_title

Bioorganic & medicinal chemistry letters

authors

Sulsky R,Robl JA,Biller SA,Harrity TW,Wetterau J,Connolly F,Jolibois K,Kunselman L

doi

10.1016/j.bmcl.2004.07.069

subject

Has Abstract

pub_date

2004-10-18 00:00:00

pages

5067-70

issue

20

eissn

0960-894X

issn

1464-3405

pii

S0960-894X(04)00971-0

journal_volume

14

pub_type

杂志文章

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