Abstract:
:A series of pyrazoline derivatives were prepared for evaluating their acyl-CoA:cholesterol acyltransferase activities. 3-(3,5-Di-tert-butyl-4-hydroxyphenyl)-5-(multi-substituted 4-hydroxyphenyl)-2-pyrazolines 4a-i were shown in vitro inhibitory activity on hACAT-1 and -2.
journal_name
Bioorg Med Chem Lettjournal_title
Bioorganic & medicinal chemistry lettersauthors
Jeong TS,Kim KS,An S,Cho KH,Lee S,Lee WSdoi
10.1016/j.bmcl.2004.03.079subject
Has Abstractpub_date
2004-06-07 00:00:00pages
2715-7issue
11eissn
0960-894Xissn
1464-3405pii
S0960894X04004524journal_volume
14pub_type
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