Discovery and in vitro evaluation of potent kinase inhibitors: Pyrido[1',2':1,5]pyrazolo[3,4-d]pyrimidines.

Abstract:

:The discovery, synthesis, potential binding mode, and in vitro kinase profile of several pyrido[1',2':1,5]pyrazolo[3,4-d]pyrimidines as potent kinase inhibitors are discussed.

journal_name

Bioorg Med Chem Lett

authors

Alberti MJ,Auten EP,Lackey KE,McDonald OB,Wood ER,Preugschat F,Cutler GJ,Kane-Carson L,Liu W,Jung DK

doi

10.1016/j.bmcl.2005.05.100

subject

Has Abstract

pub_date

2005-08-15 00:00:00

pages

3778-81

issue

16

eissn

0960-894X

issn

1464-3405

pii

S0960-894X(05)00689-X

journal_volume

15

pub_type

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