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2-(Anilino)imidazolines and 2-(benzyl)imidazoline derivatives as h5-HT1D serotonin receptor ligands.

Abstract：

:2-(Anilino)imidazolines were identified as novel human 5-HT(1D) receptor ligands, but offered no particular advantage over previously reported 2-(benzyl)imidazolines. Pharmacokinetic and functional data were obtained for selected 2-(benzyl)imidazoline derivatives.

journal_name

Bioorg Med Chem Lett

journal_title

Bioorganic & medicinal chemistry letters

authors

Prisinzano T,Dukat M,Law H,Slassi A,MacLean N,DeLannoy I,Glennon RA

doi

10.1016/j.bmcl.2004.06.085

subject

Has Abstract

pub_date

2004-09-20 00:00:00

pages

4697-9

issue

18

eissn

0960-894X

issn

1464-3405

pii

S0960-894X(04)00860-1

journal_volume

14

pub_type

杂志文章

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