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Synthesis and transacylating reactivity of beta-cyclodextrin ethylenediamines.

Abstract：

:The synthesis of the ethylenediamine-connected cyclodextrin dimer is reported, together with the syntheses of several reference cyclodextrinylamines. Each compound displayed enhanced transacylation or transphosphorylation of activated substrates, with the primary amine-bearing monocyclodextrin compound showing the greatest activity. No special rate advantage was observed for this cyclodextrin dimer, although such effects do exist in other cycloextrin dimers reported previously.

journal_name

Bioorg Med Chem

journal_title

Bioorganic & medicinal chemistry

authors

Beeson JC,Czarnik AW

doi

10.1016/s0968-0896(00)82172-0

subject

Has Abstract

pub_date

1994-04-01 00:00:00

pages

297-303

issue

4

eissn

0968-0896

issn

1464-3391

pii

S0968-0896(00)82172-0

journal_volume

2

pub_type

杂志文章

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