Abstract:
:A new method has been developed for the umpolung α-heteroarylation of ketones via an N-alkoxyenamine. The treatment of ketones with tris(heteroaryl)aluminum reagents in the presence of isoxazolidine gave the corresponding α-heteroarylated ketones in moderate to good yields.
journal_name
Chem Pharm Bull (Tokyo)journal_title
Chemical & pharmaceutical bulletinauthors
Miyoshi T,Takeda N,Fukami M,Sato S,Ueda M,Miyata Odoi
10.1248/cpb.c14-00404subject
Has Abstractpub_date
2014-01-01 00:00:00pages
927-32issue
9eissn
0009-2363issn
1347-5223pii
DN/JST.JSTAGE/cpb/c14-00404journal_volume
62pub_type
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