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Ex vivo anticholinesterase activity of benzoic acid derivatives.

Abstract：

:p-Aminobenzoic acid (p-ABA) derivatives were evaluated as acetylcholinesterase inhibitors (AChEIs). Finding a correlation between AChE activity with the partition coefficient (log P) and the highest occupied molecular orbital (HOMO) energy of the compounds.

journal_name

Chem Biol Interact

journal_title

Chemico-biological interactions

authors

Correa-Basurto J,Espinosa-Raya J,Vázquez-Alcántara I,Flores-Sandoval CA,Trujillo-Ferrara J

doi

10.1016/j.cbi.2005.10.055

subject

Has Abstract

pub_date

2005-12-15 00:00:00

pages

368-9

eissn

0009-2797

issn

1872-7786

pii

S0009-2797(05)00296-6

journal_volume

157-158

pub_type

杂志文章

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