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Microwave assisted synthesis of fragrant jasmone heterocyclic analogues.

Abstract：

:cis-Jasmone, from jasmonoid group, is an important jasmine odor fragrance compound. The syntheses of new heterocyclic analogues of jasmone were described. Five analogues of this compound were prepared under microwave irradiation and the results of the microwave assisted syntheses were compared with classical, thermally initiated reactions in solvent. Microwave reactions were carried out successfully, and reaction times were significantly reduced to a few minutes. Three of five obtained analogues, pyrrolidinone, oxazolidinone and thiazolidinone demonstrated an interesting, specific odor which was compared with floral, typical jasmine odor of jasmone.

journal_name

Eur J Med Chem

journal_title

European journal of medicinal chemistry

authors

Pawełczyk A,Zaprutko L

doi

10.1016/j.ejmech.2005.09.012

subject

Has Abstract

pub_date

2006-05-01 00:00:00

pages

586-91

issue

5

eissn

0223-5234

issn

1768-3254

pii

S0223-5234(06)00066-3

journal_volume

41

pub_type

杂志文章

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