当前位置： SCI文献检索 > BIOORGANIC & MEDICINAL CHEMISTRY LETTERS期刊下所有文献 > The solid phase synthesis of a series of tri-substituted hydantoin ligands for the somatostatin SST5 receptor.

The solid phase synthesis of a series of tri-substituted hydantoin ligands for the somatostatin SST5 receptor.

Abstract：

:A series of trisubstituted hydantoins has been prepared by a versatile solid phase route employing primary alcohols, amines and amino acids as the monomeric building blocks. Several compounds showed submicromolar affinity in binding assays at recombinant human somatostatin receptors.

journal_name

Bioorg Med Chem Lett

journal_title

Bioorganic & medicinal chemistry letters

authors

Sciciński JJ,Barker MD,Murray PJ,Jarvie EM

doi

10.1016/s0960-894x(98)00647-7

subject

Has Abstract

pub_date

1998-12-15 00:00:00

pages

3609-14

issue

24

eissn

0960-894X

issn

1464-3405

pii

S0960894X98006477

journal_volume

8

pub_type

杂志文章

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