当前位置： SCI文献检索 > BIOORGANIC & MEDICINAL CHEMISTRY期刊下所有文献 > Design, synthesis and biological evaluation of succinimide derivatives as potential mechanism-based inhibitors of human leukocyte elastase, cathepsin G and proteinase 3.

Design, synthesis and biological evaluation of succinimide derivatives as potential mechanism-based inhibitors of human leukocyte elastase, cathepsin G and proteinase 3.

Abstract：

:Structure-activity relationship study and in vitro biochemical studies with human leukocyte elastase, cathepsin G and proteinase 3 were conducted using a series of succinimide derivatives.

journal_name

Bioorg Med Chem

journal_title

Bioorganic & medicinal chemistry

authors

Groutas WC,Brubaker MJ,Chong LS,Venkataraman R,Huang H,Epp JB,Kuang R,Hoidal JR

doi

10.1016/0968-0896(95)00024-b

subject

Has Abstract

pub_date

1995-04-01 00:00:00

pages

375-81

issue

4

eissn

0968-0896

issn

1464-3391

pii

096808969500024B

journal_volume

3

pub_type

杂志文章

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