An Efficient Four-Step Approach Toward Fused Triazino[1,6-a] Quinazolines.

Abstract:

:Herein, we describe a simple, four-step process for the preparation of 1,2,3-triazino[1,6- a]quinazolin-13-ones. This method involves ring-opening, quinazoline-forming condensation, reduction, diazotization accompanied by rapid intramolecular cyclization in the last step afforded the desired products with structurally complex heterocyclic core in excellent to high yields.

authors

Sayahi MH,Baghersaei S,Goli F,Moghimi S,Mahdavi M,Firoozpour L,Shafiee A,Foroumadi A

doi

10.2174/1386207319666160202120802

subject

Has Abstract

pub_date

2016-01-01 00:00:00

pages

189-92

issue

3

eissn

1386-2073

issn

1875-5402

pii

CCHTS-EPUB-73416

journal_volume

19

pub_type

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