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Enantioselective synthesis of (+)-4-demethoxy-1,4-dimethyldaunomycinone.

Abstract：

:(+)-4-Demethoxy-1,4-dimethyldaunomycinone 1 was synthesized using a convergent approach. Here, the key tetracyclic compound 10 was assembled by way of a Diels-Alder reaction using the sugar-based diene 8 and the quinizarin-related dienophile 7.

journal_name

Bioorg Med Chem

journal_title

Bioorganic & medicinal chemistry

authors

Kotha S,Stoodley RJ

doi

10.1016/s0968-0896(01)00316-9

subject

Has Abstract

pub_date

2002-03-01 00:00:00

pages

621-4

issue

3

eissn

0968-0896

issn

1464-3391

pii

S0968089601003169

journal_volume

10

pub_type

杂志文章

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