当前位置： SCI文献检索 > BIOORGANIC & MEDICINAL CHEMISTRY LETTERS期刊下所有文献 > Solid-phase synthesis of 2,3-disubstituted indoles: discovery of a novel, high-affinity, selective h5-HT2A antagonist.

Solid-phase synthesis of 2,3-disubstituted indoles: discovery of a novel, high-affinity, selective h5-HT2A antagonist.

Abstract：

:The application of a novel solid-phase synthesis of 2,3-disubstituted indoles utilizing a carbamate indole linker is described resulting in the identification of the novel, high-affinity, selective h5-HT2A antagonist 19.

journal_name

Bioorg Med Chem Lett

journal_title

Bioorganic & medicinal chemistry letters

authors

Smith AL,Stevenson GI,Lewis S,Patel S,Castro JL

doi

10.1016/s0960-894x(00)00558-8

subject

Has Abstract

pub_date

2000-12-18 00:00:00

pages

2693-6

issue

24

eissn

0960-894X

issn

1464-3405

pii

S0960894X00005588

journal_volume

10

pub_type

杂志文章

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